Etu esi eji ọgwụ ọgwụ Telsartan?

Pin
Send
Share
Send

Ekwesịrị iji Telsartan, yana ọgwụ ndị ọzọ bụ ndị na-emegide ụdị nri angiotensin nke 2 maka ọtụtụ ọrịa, tinyere mmụba ọbara mgbali. Ngwá ọrụ a nwere ogologo oge. Mmetụta ahụ mgbe ejiri ya na-adịgide ruo awa 48. Ekwesịrị iji ngwa a mee ihe naanị dị ka dọkịta si kwuo ya na usoro ọgwụgwọ agaghị agafe ndị akọwapụtara na ntuziaka ahụ.

International Nonproprietary Aha

INN ọgwụ - Telmisartan.

ATX

Na nhazi ọkwa ATX nke mba ụwa, ọgwụ nwere koodu C09CA07.

Egosipụta iji telsartan maka ọtụtụ ọrịa, tinyere mmụba nke ọbara mgbali.

Weputara udi ya na ihe mebere ya

Akụkụ bụ isi nke ọgwụ ahụ bụ telmisartan. Ngwa ntinye aka nke Telsartan gụnyere polysorbate, magnesium stearate, meglumine, sodium hydroxide, mannitol, povidone. Enwere ụdị ọgwụ a jikọtara ọnụ. Ọgwụ Telsartan N, na mgbakwunye telmisartan, gụnyere hydrochlorothiazide.

Ọgwụ ahụ dị n'ụdị mbadamba. Dabere na usoro onodu ogwu, 40 ma obu 80 mg nke ihe eji eme ihe nwere ike idi na otu mbadamba. Mbadamba ụrọ nwere ọdịdị ya nke nwere ihe ọghọm yana usoro onunu ogwu. Ha dị ọcha. Ọpị nwere ike ịnwe mbadamba 7 ma ọ bụ 10. Na kaadiboodu, blisters 2, 3 ma ọ bụ 4 nwere ike ịnọ. Ngwakọta ọgwụ ọgwụ Telsartan AM, na mgbakwunye telsimartan, nwekwara amlodipine.

Omume ọgwụ

Omume nke Telsartan, nke bụ antigotin nke ụdị 2 angiotensin, sitere n'eziokwu ahụ na akụrụngwa a siri ike nwere ụdị nnabata a. Ihe dị n'ọrụ na-eme nhọrọ. O nwere ike wepu angiotensin site na ijikọ ya na ndị nabatara AT1.

Ọgwụ ahụ dị n'ụdị mbadamba.

Na nke a, ihe na-arụ ọrụ nke ọgwụ a enweghị aha ya na ndị ọzọ na - anabata ndị na - anabata ya. Ya mere, mgbe ị na-ewere 80 mg nke ọgwụ ahụ, itinye uche n'ọbara nke ihe ahụ na-arụ ọrụ ezuola igbochi mmetụta hypertensive nke ụdị 2 angiotensin.

N'okwu a, ọgwụ ahụ anaghị egbochi retin ma ghara itinye aka na arụ ọrụ nke ọwa ion. Na mgbakwunye, akụrụngwa a na-ebelata itinye uche nke aldosterone. Ihe dị n'ime ọgwụ a anaghị egbochi ACE, yabụ, mgbe ị na-eji Telsartan, enweghị mmetụta ndị ọ bụla na-esite na ọrụ bradykinin. Ihe ike n'ọrụ ọgwụ a anaghị emetụta obi ọnụọgụ obi. Ojiji nke ọgwụ a na-ebelata ohere mmadụ nwere ịnwụ n’arịa ndị ọrịa.

Mlọ ọgwụ

Mgbe ị na-a theụ ọgwụ ahụ, akụkụ ya dị n’ọrụ na-abanye ngwa ngwa. Bioavailability ruru 50%. Oke ọgwụ nke ọbara na-adị n’ime ụmụ nwoke na ụmụ nwanyị ka enwetara awa 3 mgbe nchịkwa gasịrị. Ọgwụ ahụ na-egbochi protein ndị dị na plasma. Metabolism nke ọgwụ na-aga n'ihu na ntinye nke glucuronic acid. A na-apụtakarị Metabolites na feces n'ime awa iri abụọ.

Ihe ngosi maka ojiji

Edebere ojiji nke Telsartan dị ka ọgwụgwọ Symptomatic maka ọrịa dị iche iche nke usoro obi, tinyere mmụba nke ọbara mgbali. Enwere ike iji ọgwụ ahụ na-emeso ndị nwere ihe ịrịba ama nke thrombosis. Ọ dị irè na ọgwụgwọ nke ndị ọrịa na-ata ahụhụ site na mmebi mmebi ischemic myocardial.

Edebere ojiji nke Telsartan dị ka ọgwụgwọ Symptomatic maka ọrịa dị iche iche nke usoro obi, tinyere mmụba nke ọbara mgbali.

Ngwá ọrụ ahụ na-enyere aka ịnagide ọbara mgbali nke bilitere na nzụlite ọnya ọnya. N'ime ihe ndị ọzọ, a na-enyekarị onye nnọchite maka ọgwụgwọ ọbara mgbali elu na ndị ọrịa na-arịa atherosclerosis nke akwara ọbara. Ọ bụrụ na ọ dị mkpa, enwere ike iji ọgwụ ahụ mee ihe na ọgwụgwọ nke ndị ọrịa nwere ọrịa shuga 2.

Ihe ngbanwe

Ekwesighi iji ọgwụ a n'ihu ọnụnọ nke anụ ahụ na-arụ ọrụ nke Telsartan. Na mgbakwunye, ịnweghị ike iji ọgwụ a gwọọ ndị ọrịa nwere ọrịa shuga 1 na-abanye insulin kwa ụbọchị. Na mgbakwunye, iji ọgwụ maka ọgwụgwọ nke ndị ọrịa nwere ọrịa nephropathy na-ewere ndị na-egbochi ACE.

Can nweghị ike iji ọgwụ a gwọọ ndị ọrịa nwere ọrịa shuga 1 nke na-agbanye insulin kwa mgbe.

Jiri nlezianya

Ọgwụgwọ na telsartan chọrọ oke ịkpachapụ anya na akwara redal stenosis. Na mgbakwunye, ndị ọrịa nwere mitral na aortic valve stenosis n'oge ọgwụgwọ na Telsartan chọrọ nlebara anya pụrụ iche site n'aka ndị ọrụ ahụ ike. Ekwesịrị ilebara hypokalemia na hyponatremia anya pụrụ iche. O kwere omume iji ọgwụ ahụ naanị n'okpuru nlekọta ndị dọkịta ma ọ bụrụ na onye ọrịa ahụ nwere akụkọ ntughari nke akụrụ.

Otu esi ewere telsartan?

E kwesịrị iwere ngwaọrụ ahụ 1 oge kwa ụbọchị, nke kachasị mma n'ụtụtụ. Iri nri anaghị emetụta nnabata nke ike ọgwụ a. Iji kpochapụ ọbara mgbali elu, a na-enye ọgwụ mbụ maka 20 mg kwa ụbọchị. N’ọdị n’ihu, enwere ike ịba ụba ọnụọgụ iri anọ ma ọ bụ 80 mg.

Na-arịa ọrịa shuga

Maka ndị ọrịa na-arịa ụdị ọrịa shuga 2, a na-edenye ọgwụ ahụ na mmalite nke 20 mg. N’ọdị n’ihu, enwere ike ịba ụba usoro ọgwụ kwa ụbọchị ruo 40 mg.

Iri nri anaghị emetụta nnabata nke ike ọgwụ a.

Nsonaazụ akụkụ nke Telsartan

Ojiji nke telsartan jikọtara ya na ọghọm nke ọtụtụ nsonaazụ. Ndị ọrịa na-enwekarị vertigo, adịghị ike, mgbu obi, yana ọrịa nrịanrịa.

Ọkpụkpụ afọ

Ojiji nke Telsartan na-edugakarị n'ọdịdị mgbu na diski diski.

Site n'akụkụ nke metabolism na nri

N'ime ndị ọrịa nwere ọrịa mellitus nke ọrịa shuga, iji telsartan nwere ike ịkpasu hypoglycemia na hyperkalemia.

Sistemụ akwara Central

Ngwá ọrụ nwere ike ime ka iro ụra hie nne. Ain nwere ike ịkụda mmụọ.

Site n'akụkụ nke sistemụ akwara dị n'etiti, enwere ike ịmetụta nsonaazụ n'ụdị nkụda mmụọ.

Site na usoro urinary

Inweta Telsartan nwere ike ibute nnukwu akwara ọdịda.

Site na sistem iku ume

Usoro ọgwụgwọ Telsartan nwere ike ibute ụkwara na mkpụmkpụ ume. Ọrịa ọrịa ngụgụ nwere ike ịmalite. N'ihi mbelata nke mgbochi ka ị na-a theụ ọgwụ ahụ, ọrịa ọrịa akụkụ okuku ume nwere ike ịmalite.

Na anụahụ

N'oge ọgwụgwọ na Telsartan, a na-ahụkarị mmepe nke hyperhidrosis na ndị ọrịa.

Site na usoro mkpụrụ ndụ ihe nketa

Patientsfọdụ ndị ọrịa na-ebute cystitis. N'ọnọdụ ndị a na - adịghị ahụkebe, megide nzụlite nke ọrịa na - efe efe nke mkpụrụ ndụ, sepsis nwere ike ime.

Patientsfọdụ ndị ọrịa na-ebute cystitis.

Site na usoro akwara obi

Site na ọgwụgwọ na Telsartan, ọnụọgụ obi nwere ike ịrị elu. Enwere ike ịmalite bradycardia na iwetulata ọbara mgbali elu. Na mgbakwunye, anaemia nwere ike ịmalite.

Site na usoro akwara na uru ahụ

Mgbe ị na-emeso Telsartan, azụ mgbu na mgbu azụ nwere ike ime. Na mgbakwunye, ọgụ myalgia na arthralgia nwere ike ịda.

N'akuku nke imeju na akụkụ biliary

Ọ dị ụkọ na ọgwụgwọ Telsartan na enwere mmebi imeju na ọnya biliary.

Ọ dị ụkọ na ọgwụgwọ Telsartan na imebi imeju na-emebi.

Ahụhụ

Ọ bụrụ na onye ọrịa ahụ nwere hypersensitivity, mmeghachi omume nfụkasị ahụ nwere ike ime, gosipụtara dịka ọnya ọnya na itching, yana ede ede Quincke

Mmetụta ikike ịchịkwa usoro

Nyere ike nke ọgwụ iji mee ka iro ụra na nkụda mmụọ, a ga-elebara anya mgbe ị na-anya ụgbọala.

Ntụziaka pụrụ iche

Ndi umu nwanyi ndi na-acho ime ime n’oge adighi eme ya. Akụkụ ahụ nọ n'ọrụ na-enwe mmetụta dị njọ na ọmụmụ. Na mgbakwunye, a ga-eji ịkpachara anya na ndị nwere oke ọgụ.

Jiri n'oge ime na lactation

Usoro ọgwụgwọ nke Telsartan maka ụmụ nwanyị n'afọ atọ ọ bụla dị ime adịghị anabata. A naghị akwado ya ka ọ useụọ ọgwụ maka ara ara.

Usoro ọgwụgwọ nke Telsartan maka ụmụ nwanyị n'afọ atọ ọ bụla dị ime adịghị anabata.

Cribdebere Telsartan Childrenmụaka

Nyere na amughi nchekwa nke Telsartan maka ụmụaka na ndị na-eto eto, a naghị atụ aro ka iji ọgwụ ahụ gwọọ ndị ọrịa dị otú ahụ.

Jiri na agadi

Enwere ike iji ọgwụ ahụ gwọọ ndị agadi. N'okwu a, a chọghị ndozi usoro onunu ogwu.

Ngwa maka ọrụ ezughi oke ọrụ

A na-anabata ojiji nke telsartan na ọgwụgwọ nke ndị ọrịa nwere ọrụ mgbazinye nsogbu. Enwere ihe akaebe banyere ike ị theụ ọgwụ ahụ na ọgwụgwọ nke ndị mmadụ na-arịa usoro ọgwụgwọ ọ bụla. Nke a chọrọ nyocha nke ọma banyere ọkwa potassium na ọbara.

Jiri maka ọrụ imeju na-arụ ọrụ

Enweghị ike iji ọgwụ ahụ agwọ ọrịa nke ndị nwere ọrịa imeju, yana mgbochi nke biliary tract na cholestasis.

Enweghị ike iji ọgwụ ahụ agwọ ọrịa nke ndị nwere ọrịa imeju, yana mgbochi nke biliary tract na cholestasis.

Dodoụbiga ihe ókè nke Telsartan

N'inwe otu ụdị ọgwụ ọgwụ buru oke ibu, bradycardia na tachycardia nwere ike ịpụta. N’ọnọdụ ndị a na-adịghị ahụkebe, ọbara mgbali elu na-ebelata. N'ihe banyere ịdoụbiga mmanya ókè, a na-edenye ọgwụgwọ Symptomatic.

Mmekọrịta na ọgwụ ndị ọzọ

Mgbe ị na-ewere Telsartan n'otu oge na ọgwụ immunosuppressive, ndị na-egbochi COX-2, heparin, yana ọgwụ ndị na-egbu mmụọ, ihe ize ndụ nke ịmalite hyperkalemia na-abawanye. Ojiji ya na ọgwụ mgbochi ọgwụ na - egbochi steroidal na - ebelata mmetụta antihypertensive nke Telsartan.

Na mgbakwunye, ngwakọta nke ọgwụ antihypertensive na akwara mkpụrụedemede akaghị, gụnyere Furasemide na hydrochlorothiazide, na-abawanye ihe ize ndụ nke ịmalite ọgba aghara na nguzo mmiri-electrolyte na mbelata ọbara mgbali elu. Nchịkọta ojiji nke telsartan na lithium na-abawanye nsonaazụ nsị nke mmiri. Site na ojiji nke Telsartan na system corticosteroids, a na-ahụ mbelata mmetụta antihypertensive.

Mmanya ndakọrịta

Should ga-ajụ ị takeụ mmanya mgbe ị na-anabata Telsartan.

Should ga-ajụ ị takeụ mmanya mgbe ị na-anabata Telsartan.

Analogs

Mmechi Telsartan nke nwere ụdị ọgwụgwọ ọgwụgwọ ahụ gụnyere:

  1. Mikardis.
  2. Ndị a.
  3. Telmitarsan.
  4. Ochichi.
  5. Irbesartan.
  6. Nortian.
  7. Kandụl.
  8. Kosaaar.
  9. Gụrụ.
  10. Telpres.
Telpres bụ otu n'ime analogues nke Telsartan.
Candesar bụ otu n'ime analogues nke Telsartan.
Mikardis bụ otu n'ime analogues nke Telsartan.
Teveten bụ otu n'ime analogues nke Telsartan.

Ahịa ọgwụ na-ahapụ okwu

Enwere ike zụta ọgwụ a n'ụlọ ahịa ọgwụ site na ndenye ọgwụ.

Ọnụ ego nke telsartan

Ọnụ ego Telsartan dị na ụlọ ahịa ọgwụ sitere na 220 ruo 260 rubles.

Ọnọdụ nchekwa maka ọgwụ

Na-echekwa ọgwụ n'ụlọ okpomọkụ.

Na-echekwa ọgwụ n'ụlọ okpomọkụ.

Bọchị mmebi

Can nwere ike iji ọgwụ ahụ maka afọ 2 site na ụbọchị emepụtara.

Emeputa

Emeputara Telsartan site n'aka Dr. Reddy's Laboratories Ltd., India.

Telmisartan belatara ọnwụ
Ọgwụ ọgwụ nke ọbara mgbali elu nke ihe ọhụụ emepụtara site n'aka ndị dọkịta Tomsk

Akaebe sitere n’aka ndị dọkịta na ndị ọrịa gbasara Telsartan

Margarita, onye gbara afọ 42, Krasnodar

Mgbe m na-arụ ọrụ dị ka dibịa akwara, ana m ahụkarị ndị ọrịa nwere mkpesa nke ọbara mgbali elu. Karịsịa, nsogbu yiri nke ahụ na-eme na ndị gbara afọ 40, mgbe mmụba nke ọbara mgbali na-eduga n'ọdịdị dị mma na ọdịmma ma mepụta ihe ị ga-ele anya maka ọdịdị nnukwu ọnọdụ, gụnyere nkụchi obi. N'ọnọdụ ndị dị otú a, m na-edenyekarị Telsartan maka ndị ọrịa. Anụ ahụ na-anabata ọgwụ ọfụma ọfụma ma ọ dịghị akpasu iwe iwe. Na nke a, ọgwụ nwere akpọ hypotensive utịp.

Igor, onye gbara afọ 38, Orenburg

Ọtụtụ mgbe, m na-edegara Telsartan maka ndị ọrịa nwere mkpesa nke ọbara mgbali elu. Ọgwụ a nwere mmetụta antihypertensive dị nro. N'okwu a, ọgwụ nwere ike itinye ya na ọgwụ mgbagwoju anya. Enwere ike iji ọgwụ ahụ gbochie mmepe nke pathologies nke usoro obi. Ọgwụ a adịghị eme ka ọnọdụ ndị ọrịa na-arịa atherosclerosis nke arịa dị n'akụkụ.

Vladimir, gbara afọ 43, Rostov-on-Don

A na-atụkarị anya ka eji Telsartan mee ihe maka ndị ọrịa nwere ọbara mgbali elu nwere ọrịa akụkọ ụdị shuga 2. Ojiji nke Telsartan na ndị ọrịa dị otú a anaghị eduga n'ịdị njọ na ọnọdụ izugbe ma n'otu oge ahụ jiri nwayọ belata ọbara mgbali. Inụ ọgwụ n’ebe ndị ọrịa dị otú a na-ebelata ohere ọghọm nke ọrịa obi.

Marina, 47 dị afọ, Moscow

Nsogbu nke jumps n'ime ọbara mgbali m nwere karịa afọ 10 gara aga. N'oge a, m nwara ọtụtụ ọgwụ. Ihe dị ka afọ abụọ gara aga, dị ka dọkịta nyere ya iwu, ọ malitere ị Telụ Telsartan. Ogwu ahụ bu nzọpụta m. Otu mbadamba otu ụbọchị zuru ezu iji mee ka nrụgide ahụ dị ụbọchị niile. Ọzọkwa, ọbụlagodi na m chefuru ị theụ ọgwụ, ahụtụbeghị m mmụba dị elu na ọbara mgbali ụbọchị niile. Enwere m afọ ojuju maka ojiji nke Telsartan. Ahụghị m ihe mgbaàmà ọ bụla.

Dmitry, gbara afọ 45, St. Petersburg

Nnabata nke Telsartan malitere na nkwenye nke dibia bekee. Maka m, ọgwụ a dabara nke ọma. Ọ bụrụ na, mgbe ị na-a otherụ ọgwụ ndị ọzọ, ọbara ọbara m na-awụlikwa elu nke ukwuu, nke na-emebi ọdịmma m n'ozuzu, mgbe m Telụsịrị Telsartan, echefuru m nsogbu nke ọbara mgbali elu. Ahụghị m nsonaazụ ọ bụla site na iji ọgwụ a ruo ihe karịrị otu afọ nke iji ọgwụ a.

Tatyana, 51 afọ, Murmansk

Ọbara mgbali elu na-enye m nsogbu kemgbe afọ iri na ise. Ejiri m ọgwụ dị iche iche na njikọ ha dịka ndị dọkịta gwara m, mana nsonaazụ ya anaghị adịte oge. Ihe dị ka afọ 1.5 gara aga, ọkà mmụta banyere akwara nyere Telsartan iwu. Ana m a thisụ ọgwụ a kwa ụbọchị ruo ugbu a. Afọ ojuju juru afọ. Nrụgide a akwụsiri ike, ọnweghị nkwanye ugwu. Enweghị mmetụta ọ bụla a hụrụ.

Pin
Send
Share
Send