Lozap 50 bụ ọgwụ edepụtara maka ndị ọrịa nwere ọrịa CCC.
International Nonproprietary Aha
Losartan.
ATX
Koodu ATX bu C09C A01.
Ha weputara udi ya na ihe mebere ya
Ọgwụ dị n'ụdị mbadamba ihe mkpuchi-fim. Mbadamba ụrọ nke ọ bụla nwere 50 mg nke ihe eji arụ ọrụ. Ihe kachasị dị mkpa nke ọgwụ ahụ bụ losartan.
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Ọgwụ ahụ dị n'ụdị mbadamba ihe mkpuchi-fim, mbadamba ọ bụla nwere 50 mg nke ihe ndị na-arụ ọrụ.
Mbadamba ụrọ nke nwere ihe mejupụtara nke 12.5 mg na-erekwa ere. Mbadamba ụcha ahụ na-acha ọcha na agba, ọdịdị biconvex nke ukwuu.
Omume ọgwụ
Losartan bụ ihe jikọrọ ndị na-anabata ya na angiotensin II. Ọ na-arụ ọrụ n'ụdị nnabata nke AT1; ndị na-anabata ndị na-anabata angiotensin anaghị ejikọ ọnụ.
Akụkụ ike nke ọgwụ ahụ anaghị egbochi ọrụ nke enzymes na-emetụta ntụgharị nke angiotensin nke m ka angiotensin II. A na - enyocha iwu ọbara mgbali elu site na ibelata ọkwa nke aldosterone na adrenaline na ọkwa ọbara. Onweghi mgbanwe n’ogidi nke angiotensin II n’ime ọbara.
N'okpuru mmetụta nke Lozap, iguzogide arịa ọbara ọbara na-ebelata. Ngwá ọrụ na-ebelata nrụgide na akwara akwara akwara, na-eso akpata mmụba na diuresis.
Mbelata nke mbubata ya na akwara gbasara obi na-egbochi mmepe nke mgbanwe mgbanwe hypertrophic na myocardium. Losartan na-ebelata ibu dị na obi n'oge a na-emega ahụ na ndị ọrịa na-arịa ọrịa na-adịghị ala ala nke usoro obi.
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Lozap 50 bụ ọgwụ edepụtara maka ndị ọrịa nwere ọrịa nke usoro obi.
Thisakingụ ọgwụ a esoghị nsogbu nke bradykinin. Mmetụta ndị na-achọghị ka ejikọta ya na usoro a anaghị eme n'oge ọgwụgwọ Lozap. N'ihi eziokwu ahụ bụ na anaghị egbochi ọrụ nke enzyme angiotensin na-agbanwe, a na-ebelata ọnọdụ angioedema na mmeghachi omume ndị ọzọ dị ize ndụ.
Mmetụta antihypertensive nke ọgwụ ahụ kacha egosipụta onwe ya awa 6 ka ị takingụ ọgwụ ahụ. A na-ahụzi mmetụta ahụ na-esote ụbọchị, jiri nwayọ belata.
Lozap gosipụtara ịdịmma kachasị mgbe nchịkwa na-aga n'ihu maka otu ọnwa ma ọ bụ karịa. N'okwu a, usoro ọgwụgwọ na-esobelata mpụta nke protein protein na immunoglobulins G na mmamịrị n'ime ndị ọrịa na-arịa ọrịa shuga mellitus.
Ọgwụ a na-eduga na nkwụsi ike nke mkpokọta urea na plasma. Ọ naghị emetụta mmegharị ahụ nke sistemụ akwara autonomic. Mgbe etinyere ya n'ọtụtụ ọkọlọtọ, ọ naghị agbanwe ọkwa suga.
Mlọ ọgwụ
Mwepu nke ihe ndị na - arụ ọrụ nke ihe ahụ na - arụ ọrụ na - apụta na obere eriri afọ. N'ime ụzọ mbido site na traktị hepatobiliary, ọ nwere ike ịnwe mgbanwe mgbanwe metabolic. Ihe cytochrome CYP2C9 isoenzyme na-etinye aka na usoro a. N'ihi mmekorita kemịkal, etinyere metabolite na-arụ ọrụ. Ihe ruru 15% nke ọgwụ a na-atụgharị na-agbanwe.
Ogologo bioavailability nke ihe na-arụ ọrụ dị ntakịrị karịa 30%. A na-ahụkarị ndọta plasma kachasị dị mma otu elele mgbe nchịkwa ọnụ. A na-enweta ihe ngosi yiri nke ahụ maka metabolite nọ n'ọrụ mgbe awa 3-4 gachara.
Akụkụ dị ike na-ejikọ peptides plasma kpamkpam. Penetration site na BBB nọ n'ogo pere mpe.
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Ndị dọkịta depụtara Lozap 50 maka ọgwụgwọ nke nkụchi obi na-adịghị ala ala.
A na-ewepụ ihe dị n'ọrụ nke ọgwụ ahụ ma eriri afọ yana akụrụ. Ndụ ndụ nke ihe na-agbanweghị agbanwe bụ ihe dị ka awa 2, ihe ngosi yiri ya maka metabolite nọ n'ọrụ bụ site na 6 ruo 9 awa.
Ihe achoro maka
Edere Lozap n'ọnọdụ ndị a:
- ya na obara mgbali di nkpa;
- iji belata ihe ize ndụ nke ịmalite ọrịa CVD na ndị mmadụ na-arịa ọbara mgbali elu;
- na nephropathy na-esite n'ọrịa metabolism na ọrịa ọrịa mellitus na-abụghị insulin na-akpata;
- maka ọgwụgwọ nke ọrịa obi na-adịghị ala ala.
Ihe ngbanwe
Ihe mgbochi iji ọgwụ a bụ:
- ịgwọ ọrịa mmadụ n'ọrụ ma ọ bụ ihe ndị ọzọ mejupụtara ya;
- ngwakọta nke ọgwụ na aliskiren n'ihu ọnya afọ ma ọ bụ ọdịda akụrụ;
- oge nke gest;
- oge lactation;
- afọ ụmụaka ruo afọ 18 (nhọpụta enwere ike n'ọnọdụ ụfọdụ).
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Ekwesịrị ịkpachara anya mgbe ị na-ewere Lozap 50 n'oge ọrịa obi.
Jiri nlezianya
Ekwesịrị ịdọ aka na ntị mgbe ị na-a theụ ọgwụ ahụ na ndị ọrịa nwere:
- hyperkalemia
- obi nkoropụ tinyere nnukwu akụrụ gbasara akwara;
- ọghọm nke ụbụrụ;
- nnukwu nkụchi obi na obi obi arrhythmias;
- akwara nke stasosis akwara;
- akwara obi;
- hypotension akwara;
- stenosis nke mitral na aortic valve;
- hypertrophic cardiomyopathy;
- mbelata nke olu nke inye ọbara;
- aldosteronism nke mbụ;
- ọgba aghara na nguzo mmiri-electrolyte.
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Ekwesịrị ịsa anya na mgbe ị na-a theụ ọgwụ ahụ na ndị ọrịa nwere ọrịa ụbụrụ.
Uzo esi ewere Lozap 50
A na-ewere mbadamba okwu ọnụ, n'agbanyeghị oge nri. Nchikota nke ogwu na ogwu ndi ozo nke wedata obara mgbali elu bu omume.
Standardzọ ị standardụ ọgwụ ọ forụ forụ maka ndị ọrịa na-enweghị ọrịa concomitant pathologies bụ 50 mg. A na-a drugụ ọgwụ ahụ kwa ụbọchị 1 oge kwa ụbọchị. A na-ahụkarị mmetụta hypotensive site na iji Lozap oge niile ihe dị ka ọnwa 1.
Ọ bụrụ na ọ dị mkpa, ọ ga-ekwe omume ịbawanye ọgwụ kwa ụbọchị ruo 100 mg. Ndi n’enwe ike n’igogharia olu obara na anata ọkara odika. Ndị ọrịa nwere obere akụrụngwa na-achọkwa mbelata usoro onunu ogwu.
Na nkụda obi na-adịghị ala ala, a na-atụ aro ịmalite usoro ọgwụgwọ site na iji ọgwụ 12.5 mg. Site na arụmọrụ ezughi oke, ọ nwere ike ịbawanye kwa izu asaa. Ọnụ ego ọgwụ a riri ga-abụrịrị nke na ọ ga-enwe ntighari n'etiti ịdị mma nke ọgwụgwọ yana enweghị mmeghachi omume ojoo.
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A na-ewere mbadamba okwu ọnụ, n'agbanyeghị oge nri.
Na-a drugụ ọgwụ maka ọrịa shuga
Ndị ọrịa nwere ọrịa mellitus na-abụghị insulin na-amalite ọgwụgwọ na usoro onunu ogwu. Ikekwe mmụba ya na 100 mg / ụbọchị. Njikọ ya na insulin na ụzọ ndị ọzọ iji chịkwaa ọbara shuga, ọnya anaghị abawanye ihe ize ndụ nke nsonaazụ.
Nsonaazụ
Ọkpụkpụ afọ
Ọkpụkpụ digesive nwere ike ịzaghachi ọgwụgwọ:
- ọdịdị mgbu na mpaghara epigastric;
- ngụ iwe;
- ọgbụgbọ
- vomiting
- agụụ riri;
- eriri afọ;
- bloating;
- ụba ọrụ nke enzymes na aha.
Ahụhụ Hematopoietic
Mgbe ụfọdụ hụrụ:
- anaemia
- mbelata na haemoglobin;
- thrombocytopenia;
- eosinophilia.
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Sistemụ akwara Central
Site na ụjọ usoro nwere ike ime:
- ike ọgwụgwụ;
- Dizziness
- nsogbu ihi ụra
- ntaramahụhụ;
- Obi erughị ala
- paresthesia;
- tinnitus;
- ọnwụ nke nsụhọ;
- isi ọwụwa.
Site na usoro urinary
Mgbe ụfọdụ nsonaazụ ndị na-esote na-apụta:
- ọdịda odida;
- urinary tract na-efe efe
Site na sistem iku ume
Nwere ike ime:
- ọphu ẹphe eme iphe dụ ẹji;
- pharyngitis;
- sinusitis
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Na anụahụ
Ihe ọghọm dị na:
- erythema;
- isi nkwọcha;
- uche nke ultraviolet radieshon;
- akpụkpọ akpọnwụ;
- rashes;
- hyperhidrosis.
Site na usoro mkpụrụ ndụ ihe nketa
Nwere ike ime:
- mẹkpoo ivu;
- enweghi ike.
Site na usoro akwara obi
Nwere ike ime:
- mmụba obi;
- mmụba obi;
- orthostatic ida;
- bradycardia;
- ihe mgbu n'azụ azụ azụ;
- vasculitis;
- imi.
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Site na usoro akwara
Enwere ike ịgbakwunye ọgwụgwọ ndị a:
- lumbalgia;
- ogwe
- olu mgbu;
- nkwonkwo mgbu.
Site n'akụkụ nke metabolism
Ihe mmetụta ndị na-esonụ nwere ike ime:
- ọkwa dị elu nke potassium na plasma ọbara;
- ụba creatinine;
- hyperbilirubinemia.
Ahụhụ
Nwere ike ime:
- mmeghachi omume anaphylactic;
- angioedema;
- ihe mgbochi ụbụrụ.
Ntụziaka pụrụ iche
Mmanya ndakọrịta
A naghị atụ aro ka ị jikọta Lozap na mmanya. Mmanya na-egbu egbu nwere ike ibute ịdị irè nke ọgwụgwọ.
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A naghị atụ aro ka ị jikọta Lozap na mmanya.
Mmetụta ikike ịchịkwa usoro
Emebeghị nnyocha pụrụ iche. Ọ dị mkpa ịjụ ịrụ ọrụ ihe egwu dị mkpa chọrọ nlebara anya itinye uche n'ihe gbasara nsonaazụ yana akwara.
Jiri n'oge ime na lactation
A naghị atụ aro ka ọ kọpụta ọgwụ maka nwanyị dị ime. Enweghị data a pụrụ ịdabere na ya ma Lozap nwere mmetụta teratogenic na nwa ebu n’afọ, mana n’ihi oke ihe ọghọm nke nsonaazụ ndị ọzọ, ejighị ya n’òtù ndị ọrịa a.
Womenmụ nwanyị dị ime ịnwetara ndị na - egbochi ACE na mbụ ka ekwesịrị ịgbanye ọgwụgwọ ọzọ. Ọ dị mkpa iji dochie ọgwụ ahụ ozugbo enwere ike mgbe ịchọpụta eziokwu nke ịtụrụ ime.
Enweghị ozi banyere oke nke ihe dị arụ ọrụ na mmiri ara ehi. Enweghị data bụ ihe kpatara ịhapụ inye nwa ara na ọgwụgwọ nke Lozap nne. A ghafere nwatakịrị ahụ na nri aka nwa.
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Oge ịgba akwụkwọ Lozap ruru ụmụaka 50
A naghị atụ aro ka ọ kọpụta ọgwụ maka ọgwụgwọ ụmụaka na-erubeghị afọ 18. N'ọnọdụ ụfọdụ, enwere ike iji ọgwụ maka ọgwụgwọ ọbara mgbali elu na ụmụaka okenye karịa afọ 6. Nhọpụta nke Lozap rue oge a machibidoro iwu, n'ihi na enweghị data na nchekwa nke ọgwụ maka ndị otu a.
Mgbe etinyere umuaka ndi di aro kariri iri-ano na iri ise, onodu ubochi bu nke adult Mgbe ụfọdụ enwere ike ide ọgwụ 50 nke Lozap. Ọtụtụ mgbe, a na-enye ndị ọrịa oke ibu ahụ karịa 50 n'arọ.
Jiri na agadi
Maka ndị gbara afọ iri ise na ise, a na-atụ aro ka a belata ọgwụ ị na-eme kwa ụbọchị ruo 25 mg. A na-eme nyocha ọzọ maka ịdị irè nke ọgwụgwọ. Ọ bụrụ na ọ dị mkpa, dọkịta na-agbazi ọgwụ a.
Ngwa maka ọrụ ezughi oke ọrụ
Inweta angiotensin-inughari enzyme inhibitors nwere ike ime ka ihe mgbaàmà nke dysfunction kelia ka njọ. E gosipụtara nke a site na mmụba nke mkpokọta nke creatinine na urea n'ọbara.
Jiri maka ọrụ imeju na-arụ ọrụ
Na nkụpu imeju n'oge ọgbụgba, mgbanwe dị na mpaghara na-arụ ọrụ na plasma ga-ekwe omume.
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Jiri maka nkụchi obi
Ọkpụkpụ akwara obi na-ebute oke ọrịa hypotension siri ike na ndị ọrịa na-ewere Lozap. Ekwesịrị ịkpachara anya mgbe ị na-edegara ndị nwere ụdị nsogbu ahụ ọgwụ ahụ.
Dodoụbiga ya ókè
An anụbiga Lozap ókè, ọ̀tụ̀tụ̀ ọbara ji erugharị n'ahụ́, mmụba obi na-apụta. A na-ewepụ ọrịa site na nhọpụta nke diuretics, ọgwụgwọ Symptomatic.
Mmekọrịta na ọgwụ ndị ọzọ
Nchikota nke ọgwụ ahu na ogwu ndi ozo. Iji nkwonkwo mee ihe na ọgwụ mgbochi ọgwụ na-akwalite mmetụta hypotensive.
Ọgwụ ndị na-emetụta ọrụ CenP2C9 isoenzyme nwere ike ịbawanye ma ọ bụ belata arụmọrụ nke ọgwụgwọ. A naghị atụ aro ka jikọta nchịkwa Lozap na ọgwụ, ihe bụ isi ọrụ ya bụ ọgwụ potassium.
A naghị akwado ya ka ijikọta nchịkwa na angiotensin-na-agbanwe enzyme inhibitors.
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Nchikota nke ọgwụ ahu na ogwu ndi ozo.
Analogs
A na-eji ndị ọrụ ndị a edochi anya ọgwụ a:
- Angizap;
- Hyperzar;
- Closart;
- Cozaar;
- Xartan
- Losartan Sandoz;
- Losex;
- Lozap Plus;
- Lozap AM;
- Lorista
- Presartan;
- Pulsar
- Centor;
- Tozaar;
- Rosan;
- Erinorm.
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Ihe atụ Russia nke ọgwụ mmanụ a Loụ Lozap 50 nwere ike ịbụ ọgwụ Blocktran.
Russian analogues nke ọgwụ:
- Ngọngọ;
- Losartan Canon;
- Lortenza.
Okwu ezumike Lozapa 50 site na pharmacies
A na-ewepụta ya dị ka ọgwụ dọkịta si ede.
Enwere m ike ịzụta na ndenye ọgwụ
Ee e.
Ọnụahịa
Ọnụ ego ahụ dabere na ebe ịzụta.
Ọnọdụ nchekwa maka ọgwụ
Ekwesịrị idobe ya na okpomọkụ agaghị akarị + 30 Celsius.
Bọchị mmebi
N'okpuru ọnọdụ nchekwa, enwere ike iji ọgwụ ahụ mee ihe n'ime ọnwa 24 site na ụbọchị ntọhapụ. A naghị atụ aro iji ihe ndị ọzọ.
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Iji dochie ọgwụ Lozap 50 na-eji ọgwụ ọgwụ Presartan.
Emeputa Lozap 50
A na-emepụta ngwaahịa ahụ site n'aka ụlọ ọrụ Slovak Saneca Pharmaceuticals.
Nyocha na Lozap 50
Ndi Okacha Cardio
Oleg Kulagin, dibia bekee, Moscow
Lozap bụ ezigbo ọgwụ maka ọgwụgwọ ọbara mgbali elu. N'ihi eziokwu ahụ na nsonaazụ ya esoghị na iwepu ọrụ ACE, ọ nwere obere mmetụta ọ bụla. Ngwá ọrụ chọrọ ịkpachara anya iji. Ekwesịrị ịnwale ndị ọrịa nwere ọrụ gbasara akụrụngwa oge ka ha wee lelee ọnọdụ anụ ahụ. Azụkwala ọgwụ a n’ejighị dọkịta. Conductme ọgwụgwọ na-enweghị mmerụ ahụ ga-enyere naanị nhọta usoro ọgwụgwọ ziri ezi, nke a ga-enyefe onye ọkachamara.
Ulyana Makarova, dibia bekee, St. Petersburg
Ngwá ọrụ ahụ na-enyere aka iji ezigbo ojiji. Kpoo ikpe dị iche iche na omume ha. Otu onye nwere obara ventricular hypertrophy kpebiri ịga ọgwụ onwe ya. Ọkọlọtọ usoro enyereghị aka ijikwa ọkwa nrụgide, yabụ ọ malitere were mbadamba 3 kwa ụbọchị. Ha niile kwụsịrị na nkụchi obi, nkwụghachi na ọnwụ. Ọnọdụ ndị a adịkarịghị, mana enwere ike izere nsogbu ahụike ma ọ bụrụ na ị na-agbaso ndụmọdụ dọkịta na ntuziaka maka ojiji.
Ndị ọrịa
Ruslan, 57 afọ, Vologda
Anọ m na-a loụ losartan ọtụtụ afọ. Nsonaazụ ndị a na-adịghị ahụkebe n'oge ọgwụgwọ. A na-etinye nrụgide ahụ n'etiti oke kwesịrị, mana m ga-eme ka onodu ogwu ahụ bukwuo elu karịa. Ahụ́ ga-eji ahụ gị mee ọgwụ ọ bụla, yabụ n'oge na-adịghị anya ị ga-achọ onye nnọchi gị.
Lyudmila, dị afọ 63, Samara
Ọ na-ahụ n'ọbara site n'ọtụtụ ụzọ. Lozap eji mee ihe afọ abụọ gara aga. Ruo oge ụfọdụ, nrụgide ahụ kwụsịrị, mana wee malite ibili ọzọ. Dọkịta ji ụdị ACE inhibitor were dochie ọgwụ ahụ, m na-a withụ ya. Eleghi anya usọbọ ahụ adabaghị naanị na nke m n'ihi ọrịa ahụ, mana enweghị m ike ịkwado ya.